WAY-100635 maleate salt 98%_634908-75-1

WAY-100635 maleate salt 98%
货号：GA139124 634908-75-1

英文名：WAY-100635 maleate salt

产品订购

产品货号	容量	货期	优惠价
GA139124-100mg	100mg	准现货	询价
GA139124-25mg	25mg	准现货	询价
GA139124-5mg	5mg	准现货	询价

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产品介绍 WAY-100635马来酸盐是5-HT受体拮抗剂，IC50为0.95nM
别名 ;N-[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]-N-2-pyridinylcyclohexanecarboxamide maleate salt
生化机理 WAY-100635 maleate salt is a potent, selective and high affinity SR-2B antagonist with a pIC50 of 10.4. The affinity (pKi) of WAY-100635 maleate salt for tSR-2B is 9.5. In addition, WAY-100635 maleate salt also blocks serotonin-evoked contraction of rat isolated stomach fundus.